Palladium-Catalyzed Tandem Amination Reaction for the Synthesis of 4-Quinolones
Tiankun Zhao and Bin Xu*
*Department of Chemistry, Shanghai University, Shanghai 200444, P. R. of China, Email: xubinshu.edu.cn
T. Zhao, B. Xu, Org. Lett., 2010, 12, 212-215.
DOI: 10.1021/ol902626d
Abstract
An efficient palladium-catalyzed tandem amination approach affords functionalized 4-quinolones in very good yields from easily accessible o-haloaryl acetylenic ketones and primary amines.
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Synthesis of N-Alkyl-Substituted 4-Quinolones via Tandem Alkenyl and Aryl C-N Bond Formation
J. Shao, X. Huang, X. Hong, B. Liu, B. Xu, Synthesis, 2012, 44, 1798-1808.
Key Words
ID: J54-Y2010-3630