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Synthesis of pyrazolines

Recent Literature

A one-pot synthesis of nitrogen-containing heterocycles from alkyl dihalides and primary amines and hydrazines occurs under microwave irradiation via a simple and efficient cyclocondensation in an alkaline aqueous medium.
Y. Ju, R. S. Varma, J. Org. Chem., 2006, 71, 135-141.

Arylhydrazines regioselectively react with 3-butynol in the presence of a catalytic amount of zinc triflate to give aryl-substituted pyrazolines. The resulting products are easily oxidized in a one-pot procedure to the corresponding pyrazoles.
K. Alex, A. Tillack, N. Schwarz, M. Beller, Org. Lett., 2008, 10, 2377-2379.

A novel, efficient, and general domino reaction of 2-acylaziridines with the Huisgen zwitterions furnishes 2-pyrazolines. A possible mechanism for the domino sequence is proposed.
S.-L. Cui, J. Wang, Y.-G. Wang, Org. Lett., 2008, 10, 13-16.