100 Years of the Biginelli dihydropyridine synthesis.

C. O. Kappe, Tetrahedron, 1993, 49, 6937.

Key Words:



Recent advances in the Biginelli dihydropyrimidine synthesis. New tricks from an old dog.

C. O. Kappe, Acc. Chem. Res., 2000, 33, 879.

Key Words:
ENANTIOSELECTIVE TOTAL SYNTHESIS/CALCIUM-CHANNEL BLOCKERS/DIELS-ALDER REACTIONS/COMBINATORIAL CHEMISTRY/ACID-ESTERS/ANTIHYPERTENSIVE AGENTS/ABSOLUTE-CONFIGURATION/FLUOROUS SYNTHESIS/LIBRARY SYNTHESIS/ORGANIC-SYNTHESIS



Synthetic applications or furan Diels-Alder chemistry.

C. O. Kappe, S. S. Murphree, A. Padwa, Tetrahedron, 1997, 53, 14179.

Key Words:
RING-TRANSFER-REACTION/FUNCTIONALIZED POLYCYCLIC SYSTEMS/CYCLO-ADDITION REACTIONS/ASYMMETRIC TOTAL SYNTHESIS/DERIVATIVES NAKED SUGARS/POLAR TRANSITION-STATE/OCCURRING FUSED FURANS/HIGH-PRESSURE/4H,6H-THIENO<3,4-C>FURAN 5,5-DIOXIDE/STEREOSELECTIVE SYNTHESIS