Synthesis of N-Substituted Indole Derivatives via PIFA-Mediated Intramolecular Cyclization
Yunfei Du, Renhe Liu, Gregory Linn and Kang Zhao*
*College of Pharmaceuticals and Biotechnology, Tianjin University, 300072, PRC, Email: combinologyyahoo.com
Y. Du, R. Liu, G. Linn, K. Zhao, Org. Lett., 2006, 8, 5919-5922.
DOI: 10.1021/ol062288o (free Supporting Information)
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Various N-arylated and N-alkylated indoles and pyrrole-fused aromatic compounds were synthesized by a phenyliodine bis(trifluoroacetate) (PIFA)-mediated intramolecular cyclization.
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