Organic Chemistry Portal



Gold(III)-Catalyzed Halogenation of Aromatic Boronates with N-Halosuccinimides

Di Qiu, Fanyang Mo, Zhitong Zheng, Yan Zhang and Jianbo Wang*

*Laboratory of Bioorganic Chemistry and Molecular Engineering of Ministry of Education, College of Chemistry, Peking University, Beijing 100871, China, Email:

D. Qiu, F. Mo, Z. Zheng, Y. Zhang, J. Wang, Org. Lett., 2010, 12, 5474-5477.

DOI: 10.1021/ol102350v


AuCl3-catalyzed halogenations of aryl borononates with N-halosuccinimides enables a convenient synthesis of aromatic boronates bearing halogen substituents in the aromatic ring.

see article for more examples

Key Words

Bromination, Iodination, Arylboronates

ID: J54-Y2010-3440