Methods for the Synthesis of Substituted Azetines
Andreas N. Baumann, Michael Eisold, Arif Music, Geoffrey Haas, Yu Min Kiw and Dorian Didier*
*Department of Chemistry and Pharmacy, Ludwig-Maximilians-University, Butenandtstraße 5-13, 81377 Munich, Germany, Email: dorian.didiercup.uni-muenchen.de
A. N. Baumann, M. Eisold, A. Music, G. Haas, Y. M. Kiw, D. Didier, Org. Lett., 2017, 19, 5681-5684.
DOI: 10.1021/acs.orglett.7b02838
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Abstract
A one-pot Suzuki cross-coupling or a catalyst-free arylation enable a facile introduction of aryl and heteroaryl substituents on the azetine skeleton at the position α to the nitrogen.
see article for more examples
A. N. Baumann, M. Eisold, A. Music, D. Didier, Synthesis, 2018, 50, 3149-3160.
Parallel Approaches for the Functionalization of Thietes: α-Metalation versus C-H Activation
M. Eisold, A. Müller-Deku, F. Reiners, D. Didier, Org. Lett., 2018, 20, 4654-4658.
Key Words
ID: J54-Y2017