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Iron-Catalyzed C(sp3)-H Acyloxylation of Aryl-2H Azirines with Hypervalent Iodine(III) Reagents

Lulu Wang, Hongji Li* and Lei Wang*

*Department of Chemistry, Huaibei Normal University, Huaibei, Anhui 235000, P. R. China, Email:,

L. Wang, H. Li, L. Wang, Org. Lett., 2018, 20, 1663-1666.

DOI: 10.1021/acs.orglett.8b00442

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An iron-catalyzed C(sp3)-H acyloxylation of aryl-2H azirines with hypervalent iodine(III) reagents (HIRs) provides a wide range of monoacyloxylated 3-aryl-2H-azirines in good yields.

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Key Words

azirines, PIDA

ID: J54-Y2018