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Parallel Approaches for the Functionalization of Thietes: α-Metalation versus C-H Activation

Michael Eisold, Adrian Müller-Deku, Felix Reiners, Dorian Didier*

*Department of Chemistry and Pharmacy, Ludwig-Maximilians-University, Butenandtstraße 5-13, 81377 Munich, Germany, Email: dorian.didiercup.uni-muenchen.de

M. Eisold, A. Müller-Deku, F. Reiners, D. Didier, Org. Lett., 2018, 20, 4654-4658.

DOI: 10.1021/acs.orglett.8b01961 (free Supporting Information)



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Abstract

Two complementary paths enable the synthesis of 3,4-disubstituted thietes in good yields via α-metalation or direct C-H functionalization.

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Methods for the Synthesis of Substituted Azetines

A. N. Baumann, M. Eisold, A. Music, G. Haas, Y. M. Kiw, D. Didier, Org. Lett., 2017, 19, 5681-5684.

One-Pot Preparation of Stable Organoboronate Reagents for the Functionalization of Unsaturated Four- and Five-Membered Carbo- and Heterocycles

A. N. Baumann, M. Eisold, A. Music, D. Didier, Synthesis, 2018, 50, 3149-3160.


Key Words

S-heterocycles


ID: J54-Y2018