Palladium-Catalyzed Methylation of Aryl, Heteroaryl, and Vinyl Boronate Esters
Alexander M. Haydl, John F. Hartwig*
*Department of Chemistry, University of California, Berkeley, California 94720, United States, Email: jhartwigberkeley.edu
A. M. Haydl, J. F. Hartwig, Org. Lett., 2019, 21, 1337-1341.
A Pd-catalyzed direct methylation of aryl, heteroaryl, and vinyl boronate esters with iodomethane occurs with a remarkably broad scope and is suitable for late-stage derivatization of biologically active compounds.
see article for more examples