Palladium-Catalyzed Hydroxylation of Aryl Halides with Boric Acid
Zhi-Qiang Song and Dong-Hui Wang*
*University of Chinese Academy of Sciences, Shanghai Institute of Organic Chemistry, 345 Lingling Road, Shanghai 200032, China, Email: dhwangsioc.ac.cn
Z.-Q. Song, D.-H. Wang, Org. Lett., 2020, 22, 8470-8474.
DOI: 10.1021/acs.orglett.0c03069
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Abstract
Boric acid, B(OH)3, is an efficient hydroxide reagent in a Pd-catalyzed conversion of (hetero)aryl halides to the corresponding phenols in very good yields under mild conditions. This transformation tolerates a broad range of functional groups.
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Key Words
ID: J54-Y2020