One-Pot Synthesis of Symmetrical and Asymmetrical 3-Amino Diynes via Cu(I)-Catalyzed Reaction of Enaminones with Terminal Alkynes
Changyuan Zhang*, Huosheng Guo, Lulu Chen*, Jiantao Zhang, Mengping Guo, Xuncheng Zhu, Chan Shen and Zeng Li
*College of Chemistry and Bio-engineering, Yichun University, Yichun 336000, P.R. China,
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C. Zhang, H. Guo, L. Chen, J. Zhang, M. Guo, X. Zhu, C. Shen, Z. Li, Org. Lett., 2021, 23, 8169-8173.
DOI: 10.1021/acs.orglett.1c02848
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Abstract
An economical and efficient Cu(I)-catalyzed one-pot reaction of enaminones with terminal alkynes provides symmetrical and asymmetrical 3-amino diynes in good yield under mild conditions.
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Key Words
ID: J54-Y2021